Lomifylline

Lomifylline

SCHEMBL1649451

CC(=O)CCCCn1cnc2c1c(=O)n(C)c(=O)n2C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 3/20 1.00
MAPK1 P28482 1/20 1.00
LMNA P02545 4/20 0.72
PDE4A P27815 3/20 0.72
CYP1A2 P05177 2/20 0.72
NFKB1 P19838 2/20 0.72
ACHE P22303 2/20 0.72
PMP22 Q01453 2/20 0.72
MAPT P10636 2/20 0.72
ESR1 P03372 1/20 0.72
BLM P54132 1/20 0.72
ADORA2B P29275 9/20 0.71
SMN1; SMN2 Q16637 3/20 0.63
PDE4B Q07343 2/20 0.63
PDE4C Q08493 2/20 0.63
PDE4D Q08499 2/20 0.63
TSHR P16473 2/20 0.63
USP2 O75604 1/20 0.63
TNF P01375 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10967382 0.90 MAPK1 (0.82) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL7802032 0.90 PDE4A (0.88) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL10855428 0.89 RXFP1 (0.81) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL16120975 0.89 ADORA2B (0.88) RXFP1MAPK1LMNAACHEMAPT
SCHEMBL11458743 0.88 RXFP1 (0.79) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL4270912 0.88 RXFP1 (0.79) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL10784282 0.87 PDE4A (0.80) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL9682866 0.87 RXFP1 (0.77) RXFP1MAPK1LMNAPDE4ACYP1A2
SCHEMBL16120999 0.87 ADORA2B (0.85) RXFP1MAPK1LMNAMAPTADORA2B
SCHEMBL16121000 0.87 ADORA2B (0.85) RXFP1MAPK1LMNAMAPTADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 170 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-0564461-B1 THE USE OF ANTIBODIES TO TNF OR FRAGMENTS DERIVED THEREOF AND XANTHINE DERIVATIVES FOR COMBINATION THERAPY AND COMPOSITIONS THEREFOR CELLTECH THERAPEUTICS LTD (GB) 1997-01-02 EP claimed
EP-0305743-B1 PHARMACEUTICAL MIXTURE PREPARATION, ITS MANUFACTURE AND USE HOECHST AKTIENGESELLSCHAFT (DE) 1992-11-04 EP claimed
US-5118500-A Side effect reduction when administering a xanthine derivative HOECHST AKTIENGESELLSCHAFT (DE) 1992-06-02 US claimed
WO-1992007585-A1 THE USE OF ANTIBODIES TO TNF OR FRAGMENTS DERIVED THEREOF AND XANTHINE DERIVATIVES FOR COMBINATION THERAPY AND COMPOSITIONS THEREFOR CELLTECH LIMITED (GB) 1992-05-14 WO claimed
CN-1057390-A Contain the medicine composition of cephalosporin and xanthine derivative and their purposes HOECHST AG (DE) 1992-01-01 CN claimed
EP-0462506-A1 Pharmaceutical preparations of mixtures comprising cefotaxim and derivatives of xanthine and their use Schrinner, Elmar J., Dr. (DE) 1991-12-27 EP claimed
CN-1014024-B PROCESS FOR PREPARING PHARMACEUTICALS-FORMULATION HOECHST AG (DE) 1991-09-25 CN claimed
EP-0169466-B1 MIXTURE OF XANTHIN DERIVATIVES AND O-ACETYL-SALICYLIC ACID, OR THEIR PHARMACOLOGICALLY ACCEPTABLE SALTS, AND ITS USE HOECHST AKTIENGESELLSCHAFT (DE) 1990-04-04 EP claimed
US-4880791-A BLOOD DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1989-11-14 US claimed
EP-0305743-A2 Pharmaceutical mixture preparation, its manufacture and use HOECHST AKTIENGESELLSCHAFT (DE) 1989-03-08 EP claimed
CN-1031184-A Pharmaceutical composition and preparation thereof and application HOECHST AG (DE) 1989-02-22 CN claimed
CN-85106465-A A kind of preparation process of pharmaceutical preparation 1986-10-29 CN claimed
EP-0169466-A2 Mixture of xanthin derivatives and O-acetyl-salicylic acid, or their pharmacologically acceptable salts, and its use HOECHST AKTIENGESELLSCHAFT (DE) 1986-01-29 EP claimed
US-4189469-A Pharmaceutical compositions HOECHST AKTIENGESELLSCHAFT (DE) 1980-02-19 US claimed