SCHEMBL9683487

SCHEMBL9683487

c1ccc(-n2cc3ccsc3c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.33
WNT3A P56704 1/20 0.33
CHRNE Q04844 1/20 0.32
COMT P21964 1/20 0.32
CYP3A4 P08684 1/20 0.31
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 2/20 0.31
HPGD P15428 2/20 0.31
POLB P06746 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
EP300 Q09472 1/20 0.31
KAT2B Q92831 1/20 0.31
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455368 0.73 CYP3A4 (0.41) COMTCYP3A4ALDH1A1KDM4EHPGD
SCHEMBL9684575 0.68 ALDH1A1 (0.37) CYP3A4ALDH1A1HPGDPOLBCYP1A2
Benzothiophene SCHEMBL15227137 0.66 CTNNB1 (0.43) CTNNB1WNT3A
Benzothiophene SCHEMBL6836326 0.66 CA12 (0.41) CTNNB1WNT3AKDM4E
SCHEMBL15074596 0.66
SCHEMBL15076887 0.66
SCHEMBL15070173 0.65
Benzothiophene SCHEMBL4378682 0.64 CTNNB1 (0.46) CTNNB1WNT3A
Benzothiophene SCHEMBL28758675 0.64 CTNNB1 (0.46) CTNNB1WNT3A
SCHEMBL31486453 0.64 GPR35 (0.36) CTNNB1WNT3APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475187-A1 Naphthothiophenimines for treating neuronal disorders caused by ischemia BRISTOL-MYERS SQUIBB COMPANY (US) 1992-03-18 EP disclosed
US-5064831-A N-methyl-d-aspartate receptor antagonist BRISTOL-MYERS SQUIBB CO. (US) 1991-11-12 US disclosed