SCHEMBL9685199

SCHEMBL9685199

COC(C1CCC(n2cnc3c(N)ncnc32)C1)P(=O)(O)O

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.55
ADCY5 O95622 11/20 0.53
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
NFKB1 P19838 1/20 0.51
THPO P40225 1/20 0.51
BLM P54132 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
PI4KA P42356 3/20 0.50
PI4K2B Q8TCG2 3/20 0.50
PI4K2A Q9BTU6 3/20 0.50
PI4KB Q9UBF8 3/20 0.50
ADORA3 P0DMS8 2/20 0.50
ADORA1 P30542 2/20 0.50
ADORA2B P29275 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685206 0.88 FDPS (0.43) ADORA2AADCY5
SCHEMBL9686031 0.84 ADORA3 (0.47) ADORA2AADORA3ADORA1
SCHEMBL6045681 0.78 ADCY5 (0.62) ADORA2AADCY5CYP1A2CYP3A4NFKB1
SCHEMBL6045512 0.78 ADCY5 (0.62) ADORA2AADCY5CYP1A2CYP3A4NFKB1
SCHEMBL6045801 0.78 ADCY5 (0.62) ADORA2AADCY5CYP1A2CYP3A4NFKB1
SCHEMBL6045575 0.78 ADCY5 (0.62) ADORA2AADCY5CYP1A2CYP3A4NFKB1
SCHEMBL9684255 0.77 ADCY5 (0.72) ADORA2AADCY5PI4KAPI4K2BPI4K2A
SCHEMBL17157383 0.76 ADCY5 (0.64) ADORA2AADCY5CYP1A2CYP3A4NFKB1
SCHEMBL15743402 0.76 ADCY5 (0.64) ADORA2AADCY5CYP1A2CYP3A4NFKB1
SCHEMBL17157337 0.76 ADCY5 (0.64) ADORA2AADCY5CYP1A2CYP3A4NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468866-A1 Novel carbocyclic analogs of certain nucleosides MERRELL DOW PHARMACEUTICALS INC. (US) 1992-01-29 EP claimed
EP-0468866-A1 Novel carbocyclic analogs of certain nucleosides MERRELL DOW PHARMACEUTICALS INC. (US) 1992-01-29 EP disclosed
EP-0468119-A1 Novel carbocyclic analogs of certain nucleosides MERRELL DOW PHARMACEUTICALS INC. (US) 1992-01-29 EP disclosed