SCHEMBL9685272

SCHEMBL9685272

CC(=O)c1ccc(CCC(C)NCC(O)COc2ccccc2)s1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.63
ALDH1A1 P00352 1/20 0.63
KMT2A Q03164 1/20 0.63
ADRB3 P13945 9/20 0.54
ADRB2 P07550 8/20 0.54
ADRB1 P08588 6/20 0.54
CYP2D6 P10635 1/20 0.52
DPP4 P27487 2/20 0.47
ABCB1 P08183 2/20 0.46
MAPT P10636 1/20 0.44
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685281 1.00 MEN1 (0.63) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL9684254 0.91 MEN1 (0.61) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL9684249 0.91 MEN1 (0.61) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL9684139 0.89 MEN1 (0.57) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL11017442 0.86 KMT2A (0.64) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL9685386 0.84 MEN1 (0.67) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL9685378 0.84 MEN1 (0.67) MEN1ALDH1A1KMT2AADRB3ADRB2
SCHEMBL10730327 0.81 ADRB1 (0.46) ALDH1A1ADRB3ADRB2ADRB1CYP2D6
SCHEMBL10730335 0.81 ADRB1 (0.46) ALDH1A1ADRB3ADRB2ADRB1CYP2D6
SCHEMBL10730332 0.81 ADRB1 (0.46) ALDH1A1ADRB3ADRB2ADRB1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166218-A Antilipemic agents or antiglycemic agents HOFFMANN-LA ROCHE INC. (US) 1992-11-24 US disclosed
US-5064863-A Catabolic activity, obesity, diabetes HOFFMANN-LA ROCHE INC. (US) 1991-11-12 US disclosed
EP-0140243-A2 Phenoxypropanol amines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-05-08 EP disclosed