SCHEMBL9685451

SCHEMBL9685451

CCn1ccc2nc(N3CCCN(c4nc(N)c5cc(OC)c(OC)cc5n4)CC3)ncc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.57
ADRA2B P18089 1/20 0.57
ADRA2C P18825 1/20 0.57
ADRA1D P25100 1/20 0.57
ADRA1A P35348 1/20 0.57
ADRA1B P35368 1/20 0.57
DRD3 P35462 1/20 0.57
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686141 0.97
Hydrochloric Acid SCHEMBL9686615 0.85 ADRA1A (0.49) ADRA2CADRA1AADRA1BKCNH2
SCHEMBL9686198 0.85 TSHR (0.40)
SCHEMBL11869688 0.76 KDM4E (0.78) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL31187488 0.76 KDM4E (0.82) ADRA1AADRA1B
SCHEMBL31151021 0.75 EHMT2 (0.69) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL5137299 0.74 KDM4E (0.76) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL29393496 0.74 POLB (0.80) ADRA1AADRA1B
Hydrochloric Acid SCHEMBL9686209 0.74 POLB (0.56) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL30555731 0.74 EHMT2 (0.68) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed