SCHEMBL9685540

SCHEMBL9685540

Cc1nc2c(F)cccc2c(Cl)c1CCCl

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
KDM4E B2RXH2 2/20 0.49
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
MAPT P10636 1/20 0.43
PDE10A Q9Y233 1/20 0.36
CD38 P28907 2/20 0.35
PKM P14618 1/20 0.35
ADORA2A P29274 4/20 0.34
ADORA1 P30542 3/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2830264 0.84 ALDH1A1 (0.58) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL5826547 0.82 ALDH1A1 (0.56) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL9685516 0.79 KDM4E (0.77) ALDH1A1KDM4EKMT2AMEN1MAPT
Hydrochloric Acid SCHEMBL9684702 0.78 KDM4E (0.75) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL2838064 0.75 KDM4E (0.55) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL2833930 0.74 MAOA (0.52) ALDH1A1KDM4EKMT2APKM
SCHEMBL8444755 0.74 MAOA (0.43) ALDH1A1KDM4EKMT2AMEN1MAPT
Hydrochloric Acid SCHEMBL9686560 0.73 MAOA (0.50) ALDH1A1KDM4EKMT2APKM
SCHEMBL2123230 0.72 AURKA (0.37) ALDH1A1KDM4EPDE10AADORA2AADORA1
SCHEMBL14843245 0.70 AR (0.36) ALDH1A1KDM4EKMT2AMEN1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0307078-B1 QUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1992-08-26 EP disclosed
US-5051508-A Antisecretory agents and enzyme inhibitors as antiulcer agents SMITHKLINE BECKMAN INTERCREDIT B.V. (NL) 1991-09-24 US disclosed
EP-0307078-A1 Quinoline derivatives, process for their preparation and pharmaceutical compositions containing them SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1989-03-15 EP disclosed