SCHEMBL9685860

SCHEMBL9685860

COc1cc(NN)ncn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.50
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
KMT2A Q03164 7/20 0.43
MEN1 O00255 5/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
ALDH1A1 P00352 4/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
STAT1 P42224 1/20 0.39
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13600415 0.81 NPC1 (0.47) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL9313620 0.79 NPC1 (0.46) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL24128114 0.78 NPC1 (0.45) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL4076540 0.77 L3MBTL1 (0.42) NPC1RAB9AKDM4EMAPTKMT2A
SCHEMBL1478401 0.77 CYP2C19 (0.48) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL12883348 0.76 NPC1 (0.44) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL8346152 0.76 CYP2C19 (0.44) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL12411077 0.76 NPC1 (0.44) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL6386093 0.74 CYP2C19 (0.47) CYP2C19NPC1RAB9AKDM4EMAPT
SCHEMBL24344306 0.73 KMT2A (0.47) CYP2C19NPC1RAB9AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0313630-B1 SUBSTITUTED 2-ACYLPYRIDIN-ALPHA-(N)-HETARYLHYDRAZONES AND MEDICAMENTS CONTAINING SAME DEUTSCHES AUSSÄTZIGEN HILFSWERK E.V. (DE) 1992-09-16 EP disclosed
US-5084458-A Bactericides, malaria and antitumor agents SCHAPER KLAUS JUERGEN (DE) 1992-01-28 US disclosed
US-4997835-A Bactericides, malaria, antitumor SCHAPER KLAUS JUERGEN (DE) 1991-03-05 US disclosed
EP-0313630-A1 SUBSTITUTED 2-ACYLPYRIDIN-ALPHA-(N)-HETARYLHYDRAZONES AND MEDICAMENTS CONTAINING SAME. DEUTSCHES AUSSATZIGEN HILFSWER (DE) 1989-05-03 EP disclosed