SCHEMBL9686643

SCHEMBL9686643

CC(=O)CN1CCN(c2nc3c(cc2F)c(=O)c(C(=O)O)cn3C2CC2)CC1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.56
CHRM2 P08172 1/20 0.56
DRD1 P21728 1/20 0.56
KDM4E B2RXH2 5/20 0.52
LMNA P02545 5/20 0.52
HSD17B10 Q99714 2/20 0.52
ABCC4 O15439 1/20 0.52
DHFR P00374 1/20 0.49
ALDH1A1 P00352 4/20 0.47
CYP2C9 P11712 1/20 0.47
ATP6V1B2 P21281 1/20 0.47
TBXA2R P21731 1/20 0.47
EDNRA P25101 1/20 0.47
TARBP2 Q15633 1/20 0.47
KMT2A Q03164 1/20 0.47
HPGD P15428 2/20 0.47
MAPT P10636 1/20 0.47
TDP1 Q9NUW8 2/20 0.45
POLB P06746 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686650 0.89 DPP4 (0.46) DPP4CHRM2DRD1KDM4ELMNA
Hydrochloric Acid SCHEMBL10548709 0.86 DHFR (0.57) DPP4CHRM2DRD1KDM4ELMNA
Hydrochloric Acid SCHEMBL10549780 0.86 DPP4 (0.59) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL10920054 0.82 KDM4E (0.68) KDM4ELMNAHSD17B10ALDH1A1CYP2C9
SCHEMBL9687603 0.82 KDM4E (0.66) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL10377610 0.81 DPP4 (0.62) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL9687753 0.81 KDM4E (0.63) DPP4CHRM2DRD1KDM4ELMNA
Hydrochloric Acid SCHEMBL10557063 0.81 DHFR (0.56) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL10928412 0.81 DPP4 (0.64) DPP4CHRM2DRD1KDM4ELMNA
Hydrochloric Acid SCHEMBL10551866 0.81 DPP4 (0.61) DPP4CHRM2DRD1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4840954-A BACTERICIDE BAYER AKTIENGESELLSCHAFT (DE) 1989-06-20 US claimed
EP-0187376-B1 6,7-DISUBSTITUTED 1-CYCLOPROPYL-1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACIDS BAYER AG (DE) 1992-05-13 EP disclosed
US-4840954-A BACTERICIDE BAYER AKTIENGESELLSCHAFT (DE) 1989-06-20 US disclosed