SCHEMBL9687706

SCHEMBL9687706

CCCC(c1noc2ccccc12)n1ccnc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 13/20 0.53
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
CYP19A1 P11511 4/20 0.38
GRM4 Q14833 1/20 0.37
FAAH O00519 1/20 0.36
MGLL Q99685 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10464807 0.90 CYP17A1 (0.51) CYP17A1CYP11B1CYP11B2CYP3A4
Oxalic Acid SCHEMBL9687827 0.87 CYP17A1 (0.52) CYP17A1CYP11B1CYP11B2CYP19A1FAAH
SCHEMBL9688917 0.82 CYP17A1 (0.54) CYP17A1CYP19A1
SCHEMBL9688727 0.81 CYP17A1 (0.40) CYP17A1CYP11B1CYP11B2CYP19A1CYP3A4
SCHEMBL9689763 0.80 CYP17A1 (0.48) CYP17A1CYP11B1CYP11B2CYP19A1CYP3A4
SCHEMBL10465932 0.75 CYP17A1 (0.53) CYP17A1CYP11B1CYP11B2CYP19A1CYP3A4
SCHEMBL21678833 0.75 FAAH (0.46) GRM4FAAHMGLLCYP3A4
SCHEMBL4578052 0.74 CYP17A1 (0.83) CYP17A1CYP11B1CYP11B2CYP19A1CYP3A4
SCHEMBL20003881 0.72 GRM4 (0.49) GRM4FAAHMGLLCYP3A4
SCHEMBL21976453 0.72 FAAH (0.44) GRM4FAAHMGLLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298921-B1 1,2-BENZISOXAZOLES AND 1,2-BENZISOTHIAZOLES CIBA-GEIGY AG (CH) 1992-12-23 EP disclosed
US-4957931-A ANTICONVULSANTS, TREATMENT OF EPILEPSY CIBA-GEIGY CORPORATION (US) 1990-09-18 US disclosed
US-4859691-A Certain 1,2-benzisoxazole derivatives CIBA-GEIGY CORPORATION (US) 1989-08-22 US disclosed
EP-0298921-A1 1,2-Benzisoxazoles and 1,2-benzisothiazoles CIBA-GEIGY AG (CH) 1989-01-11 EP disclosed