SCHEMBL9687791

SCHEMBL9687791

COc1ccnc(CSc2nc3c(C)c(OC(F)F)c(C)cc3[nH]2)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 11/20 0.44
ATP4B P51164 11/20 0.44
CYP2C9 P11712 3/20 0.43
CYP3A4 P08684 3/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SLC22A2 O15244 1/20 0.43
DDAH1 O94760 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
ABCB1 P08183 1/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
ADRA1A P35348 1/20 0.43
FASN P49327 1/20 0.43
SLC47A2 Q86VL8 1/20 0.43
SLC47A1 Q96FL8 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
BRS3 P32247 1/20 0.41
CYP1A2 P05177 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686676 0.93 CYP3A4 (0.46) ATP4AATP4BCYP2C9CYP3A4HPGD
SCHEMBL9686799 0.86 CYP2C9 (0.45) ATP4AATP4BCYP2C9CYP3A4HPGD
SCHEMBL9687921 0.84 CYP1A2 (0.45) CYP2C9CYP3A4HPGDALDH1A1LMNA
SCHEMBL9687828 0.84 ATP4A (0.47) ATP4AATP4BCYP2C9CYP3A4HPGD
SCHEMBL9688506 0.84 ATP4A (0.47) ATP4AATP4BCYP2C9CYP3A4HPGD
SCHEMBL9688793 0.84 CYP3A4 (0.44) ATP4AATP4BCYP2C9CYP3A4HPGD
SCHEMBL9687805 0.83 BRS3 (0.57) ATP4AATP4BCYP2C9CYP3A4HPGD
SCHEMBL9687792 0.82 NOS2 (0.55) ATP4AATP4BCYP2C9CYP3A4BRS3
SCHEMBL9793565 0.81 BRS3 (0.53) CYP2C9CYP3A4LMNABRS3CYP1A2
SCHEMBL9688807 0.81 CYP1A2 (0.45) CYP2C9CYP3A4HPGDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201575-B1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1992-08-12 EP disclosed
US-4686230-A Picoline derivative useful as gastric acid secretion inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1987-08-11 US disclosed
EP-0093320-B1 PROCESS FOR THE EXTRACTION OF ONIUM SALTS FROM PROCESS AND WASTE WATERS BAYER AG (DE) 1987-06-16 EP disclosed
EP-0093320-A2 Process for the extraction of onium salts from process and waste waters BAYER AG (DE) 1983-11-09 EP disclosed