SCHEMBL9688984

SCHEMBL9688984

Nc1nc2cccnc2n1C1CCCNCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.57
PDE4B Q07343 3/20 0.46
PDE4D Q08499 3/20 0.46
HCAR1 Q9BXC0 1/20 0.40
PIK3CD O00329 4/20 0.39
ALDH1A1 P00352 3/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
ALOX15 P16050 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539176 0.95 TP53 (0.62) TP53PDE4BPDE4DHCAR1ALDH1A1
SCHEMBL16084474 0.88 PDE4B (0.52) TP53PDE4BPDE4DHCAR1ALDH1A1
SCHEMBL5775620 0.86 PDE4B (0.54) TP53PDE4BPDE4DHCAR1ALDH1A1
SCHEMBL5778683 0.86 PDE4B (0.54) TP53PDE4BPDE4DHCAR1ALDH1A1
SCHEMBL5775573 0.86 PDE4B (0.54) TP53PDE4BPDE4DHCAR1ALDH1A1
SCHEMBL2790752 0.79 TP53 (0.65) TP53PDE4BPDE4DPOLBALOX15
SCHEMBL12893949 0.76 TP53 (0.59) TP53PDE4BPDE4DPOLBHTR3E
SCHEMBL6160948 0.75 TP53 (0.58) TP53PDE4BPDE4DALDH1A1HSD17B10
SCHEMBL9685823 0.74 RPS6KB1 (0.47) TP53ALDH1A1MEN1MAPTPKM
SCHEMBL13319030 0.73 TP53 (0.62) TP53PDE4BPDE4DALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed