SCHEMBL9688992

SCHEMBL9688992

COc1cccc(C2C(C(=O)O)=C(C)NC(C)=C2C(=O)O)c1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
NPC1 O15118 1/20 0.54
TSHR P16473 4/20 0.49
ATM Q13315 1/20 0.48
ALDH1A1 P00352 3/20 0.47
HSD17B10 Q99714 3/20 0.47
CASP1 P29466 2/20 0.47
HPGD P15428 1/20 0.47
CASP7 P55210 1/20 0.47
BAP1 Q92560 1/20 0.47
KDM4E B2RXH2 3/20 0.47
GLA P06280 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 5/20 0.47
NR1I2 O75469 1/20 0.46
PKM P14618 1/20 0.46
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10367692 0.94 NR1I2 (0.56) GAASMN1; SMN2NPC1TSHRATM
SCHEMBL9806975 0.87 MAPT (0.56) GAASMN1; SMN2NPC1TSHRALDH1A1
SCHEMBL7414856 0.81 NR1I2 (0.67) GAASMN1; SMN2TSHRALDH1A1HSD17B10
SCHEMBL7025790 0.78 NR1I2 (0.56) GAASMN1; SMN2NPC1TSHRALDH1A1
SCHEMBL10675417 0.75 NR1I2 (0.53) GAASMN1; SMN2TSHRALDH1A1HSD17B10
SCHEMBL7106117 0.75 KDM4E (0.56) GAASMN1; SMN2TSHRALDH1A1HSD17B10
SCHEMBL9690101 0.75 KMT2A (0.43) GAATSHRATMALDH1A1HSD17B10
SCHEMBL10596292 0.74 GAA (0.54) GAASMN1; SMN2NPC1TSHRALDH1A1
SCHEMBL3034560 0.74 NR1I2 (0.73) GAASMN1; SMN2TSHRALDH1A1HSD17B10
SCHEMBL29676206 0.74 NR1I2 (0.73) GAASMN1; SMN2TSHRALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0158211-B1 1,4-DIHYDROPYRIDIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USES AS MEDICAMENTS LABORATORIOS DELAGRANGE S.A. (ES) 1992-08-26 EP disclosed
US-4722931-A MUSCLE RELAXANTS LABORATORIOS DELAGRANGE (ES) 1988-02-02 US disclosed
EP-0158211-A2 1,4-Dihydropyridin derivatives, process for their preparation and their uses as medicaments LABORATORIOS DELAGRANGE S.A. (ES) 1985-10-16 EP disclosed