SCHEMBL9690101

SCHEMBL9690101

COc1cc(C2C(C(=O)O)=C(C)NC(C)=C2C(=O)O)cc(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.43
ATM Q13315 1/20 0.43
KDM4E B2RXH2 4/20 0.43
LMNA P02545 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
TSHR P16473 1/20 0.42
TPMT P51580 1/20 0.41
GAA P10253 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPT P10636 1/20 0.41
RECQL P46063 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 1/20 0.41
HSD17B10 Q99714 2/20 0.41
HTR1A P08908 1/20 0.41
HTR2C P28335 1/20 0.41
CACNA1B Q00975 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690085 0.89 PKM (0.51) KDM4ELMNAALDH1A1HPGDTSHR
SCHEMBL9473905 0.83 ALDH1A1 (0.51) ATMKDM4ELMNAALDH1A1HPGD
SCHEMBL9688157 0.81 KDM4E (0.49) KDM4ELMNAALDH1A1HPGDTSHR
SCHEMBL9869972 0.78 ATM (0.43) KMT2AATMKDM4ELMNAALDH1A1
SCHEMBL11709161 0.76 GAA (0.54) ATMKDM4ELMNAALDH1A1HPGD
SCHEMBL11801987 0.76 GAA (0.54) KMT2AATMKDM4ELMNAALDH1A1
SCHEMBL9688992 0.75 GAA (0.54) ATMKDM4EALDH1A1HPGDTSHR
SCHEMBL27517088 0.74 KDM4E (0.68) KMT2AKDM4ELMNAALDH1A1HPGD
SCHEMBL9870900 0.73 ATM (0.45) KMT2AATMKDM4ELMNAALDH1A1
SCHEMBL10564440 0.73 CACNA1F (0.61) KDM4EALDH1A1HPGDGAACACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0158211-B1 1,4-DIHYDROPYRIDIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USES AS MEDICAMENTS LABORATORIOS DELAGRANGE S.A. (ES) 1992-08-26 EP disclosed
US-4722931-A MUSCLE RELAXANTS LABORATORIOS DELAGRANGE (ES) 1988-02-02 US disclosed
EP-0158211-A2 1,4-Dihydropyridin derivatives, process for their preparation and their uses as medicaments LABORATORIOS DELAGRANGE S.A. (ES) 1985-10-16 EP disclosed