SCHEMBL9689496

SCHEMBL9689496

CCN(CC)c1ccc([N+](=O)[O-])c(N2CCNCC2)n1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.46
ALDH1A1 P00352 6/20 0.46
MAPK1 P28482 3/20 0.46
POLB P06746 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
RECQL P46063 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTR6 P50406 1/20 0.41
ADRB1 P08588 1/20 0.40
SIRT6 Q8N6T7 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745501 0.82 MAPT (0.43) MAPTALDH1A1MAPK1POLBTDP1
SCHEMBL8547098 0.79 HRH4 (0.38) ALDH1A1
SCHEMBL6284789 0.79 MAPT (0.52) MAPTALDH1A1MAPK1POLBTDP1
SCHEMBL9069903 0.78 HRH4 (0.42) ALDH1A1SMN1; SMN2
SCHEMBL9069901 0.78 ALDH1A1 (0.48) MAPTALDH1A1MAPK1POLBTDP1
SCHEMBL9073188 0.76 KDM4E (0.38) MAPTSMN1; SMN2HTR6CYP1A2CYP2C19
SCHEMBL952111 0.76 POLB (0.58) MAPTALDH1A1MAPK1POLBTDP1
Diethylamine SCHEMBL10719828 0.73 CCNT1 (0.35) ALDH1A1
Diethylamine SCHEMBL10365487 0.72 HRH4 (0.39) ALDH1A1SMN1; SMN2
SCHEMBL2982554 0.72 MAPT (0.43) MAPTALDH1A1MAPK1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
US-4996318-A Amino-9,10-secosteroids useful for treating head injury, spinal cord trauma or stroke THE UPJOHN COMPANY (US) 1991-02-26 US disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0354920-A1 AMINO-9,10-SECOSTEROIDS THE UPJOHN COMPANY (US) 1990-02-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed
WO-1988007527-A1 AMINO-9,10-SECOSTEROIDS THE UPJOHN COMPANY (US) 1988-10-06 WO disclosed
EP-0263213-A1 C20 Through C26 amino steroids THE UPJOHN COMPANY (US) 1988-04-13 EP disclosed
EP-0238545-A1 C 20? THROUGH C 26? AMINO STEROIDS. UPJOHN CO (US) 1987-09-30 EP disclosed
WO-1987001706-A2 C20 THROUGH C26 AMINO STEROIDS THE UPJOHN COMPANY (US) 1987-03-26 WO disclosed