SCHEMBL9689545

SCHEMBL9689545

CCOC(=O)OC1=C(C)NC2=C(C(=O)OC2)C1c1cccc(Cl)c1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
KDM4E B2RXH2 4/20 0.52
CYP2C9 P11712 3/20 0.48
TSHR P16473 3/20 0.48
GAA P10253 3/20 0.48
MEN1 O00255 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C19 P33261 2/20 0.48
KMT2A Q03164 2/20 0.48
HIF1A Q16665 2/20 0.48
HSD17B10 Q99714 2/20 0.48
ABCB11 O95342 2/20 0.48
LMNA P02545 2/20 0.48
MAPT P10636 2/20 0.48
HPGD P15428 1/20 0.48
TP53 P04637 1/20 0.48
CYP2D6 P10635 1/20 0.48
NFKB1 P19838 1/20 0.48
THPO P40225 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10648966 0.92 ALDH1A1 (0.56) ALDH1A1KDM4ECYP2C9TSHRGAA
SCHEMBL11008190 0.86 KDM4E (0.67) ALDH1A1KDM4ECYP2C9TSHRGAA
SCHEMBL9690702 0.86 KDM4E (0.53) ALDH1A1KDM4ETSHRGAAMEN1
SCHEMBL9690787 0.86 ALDH1A1 (0.58) ALDH1A1KDM4ETSHRGAAMEN1
SCHEMBL10652934 0.85 ALDH1A1 (0.51) ALDH1A1KDM4ETSHRGAAKMT2A
SCHEMBL9692020 0.85 ALDH1A1 (0.57) ALDH1A1KDM4ECYP2C9TSHRGAA
SCHEMBL9839402 0.85 ALDH1A1 (0.57) ALDH1A1KDM4ETSHRGAAMEN1
SCHEMBL9689704 0.82 KDM4E (0.57) ALDH1A1KDM4ETP53CACNA1FCACNA1D
SCHEMBL9691494 0.82 ALDH1A1 (0.54) ALDH1A1KDM4ETSHRGAAMEN1
SCHEMBL9689623 0.82 ALDH1A1 (0.57) ALDH1A1KDM4EGAAMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed