SCHEMBL9689611

SCHEMBL9689611

CCOC(=O)OC1=C(C)NC2=C(C(=O)OC2)C1c1ccccc1SCc1cccc([N+](=O)[O-])c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CACNA1C Q13936 9/20 0.40
MEN1 O00255 3/20 0.40
MAPT P10636 3/20 0.40
KMT2A Q03164 3/20 0.40
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
CACNA1F O60840 7/20 0.39
CACNA1D Q01668 7/20 0.39
CACNA1S Q13698 7/20 0.39
ADORA3 P0DMS8 2/20 0.39
HIF1A Q16665 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691280 0.92 ALDH1A1 (0.45) ALDH1A1KDM4ECACNA1CMEN1MAPT
SCHEMBL11006153 0.89 ALDH1A1 (0.54) ALDH1A1KDM4ECACNA1CMEN1MAPT
SCHEMBL9691845 0.89 ALDH1A1 (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL9691606 0.88 KDM4E (0.52) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL11008399 0.86 ALDH1A1 (0.46) ALDH1A1KDM4ECACNA1CMEN1MAPT
SCHEMBL11008396 0.86 ALDH1A1 (0.46) ALDH1A1KDM4ECACNA1CMEN1MAPT
SCHEMBL10817896 0.85 ALDH1A1 (0.48) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL9691203 0.85 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTKMT2AGAA
SCHEMBL9689606 0.84 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL9689646 0.84 KDM4E (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed