SCHEMBL11006153

SCHEMBL11006153

CCOC(=O)C1=C(C)NC2=C(C(=O)OC2)C1c1ccccc1SCc1cccc([N+](=O)[O-])c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 1/20 0.54
CACNA1C Q13936 11/20 0.49
CACNA1F O60840 10/20 0.49
CACNA1D Q01668 10/20 0.49
CACNA1S Q13698 10/20 0.49
ADORA3 P0DMS8 2/20 0.49
HIF1A Q16665 3/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
MAPT P10636 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 1/20 0.49
MAPK1 P28482 1/20 0.49
GPR55 Q9Y2T6 1/20 0.49
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11006991 0.91 ALDH1A1 (0.57) ALDH1A1KDM4ECACNA1CCACNA1FCACNA1D
SCHEMBL11008399 0.91 ALDH1A1 (0.46) ALDH1A1KDM4ECACNA1CADORA3MEN1
SCHEMBL11008396 0.91 ALDH1A1 (0.46) ALDH1A1KDM4ECACNA1CADORA3MEN1
SCHEMBL9689611 0.89 ALDH1A1 (0.43) ALDH1A1KDM4ECACNA1CCACNA1FCACNA1D
SCHEMBL11007725 0.89 KDM4E (0.59) ALDH1A1KDM4EADORA3MEN1KMT2A
SCHEMBL8803276 0.88 KDM4E (0.67) ALDH1A1KDM4EADORA3MEN1KMT2A
SCHEMBL8602349 0.88 KDM4E (0.67) ALDH1A1KDM4EADORA3MEN1KMT2A
SCHEMBL11005127 0.84 KDM4E (0.62) ALDH1A1KDM4EMAPTLMNAPOLB
SCHEMBL11005169 0.84 KDM4E (0.58) ALDH1A1KDM4ECACNA1CCACNA1FCACNA1D
SCHEMBL11007569 0.84 KDM4E (0.59) ALDH1A1KDM4EMAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4532248-A Administering 1,4-dihydropyridine derivative exhibiting positive inotropic activity BAYER AKTIENGESELLSCHAFT (DE) 1985-07-30 US disclosed