SCHEMBL9689685

SCHEMBL9689685

N=C(N)NCCCCCCC(=O)NCC(=O)NCCCCNCCCN

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 2/20 0.48
PAOX Q6QHF9 1/20 0.47
HDAC6 Q9UBN7 3/20 0.44
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
CA12 O43570 2/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA6 P23280 2/20 0.40
CA5A P35218 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
CA5B Q9Y2D0 2/20 0.40
ITGB3 P05106 2/20 0.40
ITGA2B P08514 2/20 0.40
CA1 P00915 1/20 0.40
CA3 P07451 1/20 0.40
HDAC3 O15379 2/20 0.39
HDAC4 P56524 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10641540 1.00 SLC6A5 (0.48) SLC6A5PAOXHDAC6MAOAMAOB
Hydrochloric Acid SCHEMBL10642172 0.99 SLC6A5 (0.49) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL11015199 0.93 PAOX (0.51) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL11011464 0.93 PAOX (0.51) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL11009412 0.91 PAOX (0.50) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL10641835 0.91 PAOX (0.50) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL524729 0.87 MAOA (0.44) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL524298 0.87 MAOA (0.44) SLC6A5PAOXHDAC6MAOAMAOB
SCHEMBL524786 0.85 PAOX (0.47) PAOXHDAC6MAOAMAOBCA12
SCHEMBL525137 0.85 PAOX (0.47) PAOXHDAC6MAOAMAOBCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4529549-A Compound containing guanidine and amino groups ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1985-07-16 US claimed
JP-59042356-A None JP disclosed
WO-2010028389-A1 IMAGE-GUIDED ENERGY DEPOSITION FOR TARGETED DRUG DELIVERY THE METHODIST HOSPITAL RESEARCH INSTITUTE (US) 2010-03-11 WO disclosed
EP-0181592-B1 USE OF SPERGUALIN DERIVATIVES FOR THE PREPARATION OF MEDICAMENTS HAVING IMMUNOSUPPRESSIVE ACTIVITY MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1992-09-16 EP disclosed
US-4851446-A SPERGUALIN-LIKE GUANIDINES ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1989-07-25 US disclosed
EP-0105193-B1 SPERGUALIN-RELATED COMPOUNDS, PROCESSES FOR THE PREPARATION THEREOF AND THEIR USE AS MEDICAMENTS MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1988-08-24 EP disclosed
EP-0181592-A2 Use of spergualin derivatives for the preparation of medicaments having immunosuppressive activity MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1986-05-21 EP disclosed
US-4529549-A Compound containing guanidine and amino groups ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1985-07-16 US disclosed
EP-0105193-A2 Spergualin-related compounds, processes for the preparation thereof and their use as medicaments MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1984-04-11 EP disclosed
JP-S5942356-A SPERGUALIN-RELATED COMPOUND AND PREPARATION THEREOF MICROBIAL CHEM RES FOUND 1984-03-08 JP disclosed