SCHEMBL9690289

SCHEMBL9690289

Cc1c(C)c2c(c(C)c1O)CCC(C)(C(=O)NCCCCc1ccccc1)O2

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 18/20 0.63
BCHE P06276 17/20 0.63
PTGS1 P23219 1/20 0.57
PTGS2 P35354 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
TSHR P16473 1/20 0.57
MAOB P27338 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690224 0.97 ACHE (0.61) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2058864 0.93 PTGS1 (0.60) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2059491 0.87 PTGS1 (0.62) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2058855 0.83 PTGS1 (0.62) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL9314334 0.82 PTGS1 (0.61) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2059279 0.82 PTGS1 (0.61) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2059293 0.82 PTGS1 (0.61) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2059199 0.82 PTGS1 (0.61) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL2058872 0.82 PTGS1 (0.64) ACHEBCHEPTGS1PTGS2CYP1A2
SCHEMBL9689071 0.82 ALOX5 (0.48) ACHEBCHEPTGS1PTGS2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP claimed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed