SCHEMBL9691124

SCHEMBL9691124

CCCN1C(C)=C(OC(=O)OCC)C(c2ccccc2SCc2ccccc2)C2=C1COC2=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.32
HTT P42858 2/20 0.31
LMNA P02545 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
BRD4 O60885 1/20 0.31
BRDT Q58F21 1/20 0.31
TRPC5 Q9UL62 1/20 0.31
NPC1 O15118 3/20 0.31
RAB9A P51151 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TSHR P16473 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30
ADORA2A P29274 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691603 0.93 ALDH1A1 (0.36) ALDH1A1KDM4EHTTLMNANPSR1
SCHEMBL9691805 0.91 ALDH1A1 (0.36) ALDH1A1KDM4EHTTLMNANPSR1
SCHEMBL9691486 0.90 ALDH1A1 (0.34) ALDH1A1KDM4EGPBAR1KMT2A
SCHEMBL11012109 0.87 ALDH1A1 (0.40) ALDH1A1KDM4EGPBAR1HTTLMNA
SCHEMBL9691774 0.83 MAPT (0.38) ALDH1A1HTTLMNANPSR1RAB9A
SCHEMBL9691700 0.81 KDM4E (0.39) ALDH1A1KDM4ENPSR1KMT2AL3MBTL1
SCHEMBL11012203 0.80 ALDH1A1 (0.41) ALDH1A1KDM4EGPBAR1HTTLMNA
SCHEMBL9691606 0.80 KDM4E (0.52) ALDH1A1KDM4EHTTLMNANPSR1
SCHEMBL11003915 0.79 KDM4E (0.45) ALDH1A1KDM4EHTTNPSR1TRPC5
SCHEMBL9691218 0.79 ALDH1A1 (0.45) ALDH1A1KDM4EHTTLMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed