SCHEMBL9691603

SCHEMBL9691603

CCOC(=O)OC1=C(C)N(CC)C2=C(C(=O)OC2)C1c1ccccc1SCc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 3/20 0.33
TSHR P16473 2/20 0.33
LMNA P02545 2/20 0.33
TRPC5 Q9UL62 1/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
KMT2A Q03164 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
ADORA2A P29274 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
MYC P01106 1/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691124 0.93 ALDH1A1 (0.35) ALDH1A1KDM4EHTTTSHRLMNA
SCHEMBL9691486 0.91 ALDH1A1 (0.34) ALDH1A1KDM4EKMT2AMEN1
SCHEMBL9691805 0.91 ALDH1A1 (0.36) ALDH1A1KDM4EHTTTSHRLMNA
SCHEMBL9691774 0.89 MAPT (0.38) ALDH1A1HTTTSHRLMNARAB9A
SCHEMBL11012203 0.87 ALDH1A1 (0.41) ALDH1A1KDM4EHTTTSHRLMNA
SCHEMBL8804777 0.85 PYGM (0.37) ALDH1A1KDM4EHTTLMNAKMT2A
SCHEMBL10649530 0.83 PYGL (0.39) ALDH1A1KDM4EHTTTSHRLMNA
SCHEMBL9691606 0.82 KDM4E (0.52) ALDH1A1KDM4EHTTTSHRLMNA
SCHEMBL9689389 0.81 KDM4E (0.40) ALDH1A1KDM4EKMT2AL3MBTL1NPSR1
SCHEMBL11012109 0.80 ALDH1A1 (0.40) ALDH1A1KDM4EHTTTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed