SCHEMBL9691675

SCHEMBL9691675

CC1=C(OC(=O)O)C(c2ccccc2OCc2ccc(C)cc2)C(OC(=O)OC(C)C)=C(C)N1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.40
SLC1A5 Q15758 1/20 0.39
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
KDM4E B2RXH2 3/20 0.36
KMT2A Q03164 3/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 2/20 0.36
GAA P10253 1/20 0.35
AKR1C3 P42330 1/20 0.35
NR1I2 O75469 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691403 0.92 TP53 (0.40) TP53SLC1A5POLBSMN1; SMN2GPBAR1
SCHEMBL9691648 0.91 TP53 (0.41) TP53SLC1A5POLBSMN1; SMN2RXRA
SCHEMBL10814309 0.91 TP53 (0.45) TP53SLC1A5POLBSMN1; SMN2RXRA
SCHEMBL10818189 0.90 TP53 (0.41) TP53SLC1A5POLBSMN1; SMN2GPBAR1
SCHEMBL10646454 0.88 POLB (0.41) TP53POLBSMN1; SMN2GPBAR1SIRT1
SCHEMBL9691359 0.86 POLB (0.44) TP53POLBSMN1; SMN2SIRT1KDM4E
SCHEMBL10649425 0.86 POLB (0.40) TP53POLBSMN1; SMN2GPBAR1SIRT1
SCHEMBL10646808 0.85 POLB (0.39) TP53POLBSMN1; SMN2GPBAR1SIRT1
SCHEMBL9691625 0.84 NR1I2 (0.42) SLC1A5POLBSMN1; SMN2SIRT1KDM4E
SCHEMBL9691661 0.84 TP53 (0.43) TP53SLC1A5POLBSMN1; SMN2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed