SCHEMBL9691625

SCHEMBL9691625

COC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.42
HTR1A P08908 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.40
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PLA2G1B P04054 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC1A5 Q15758 1/20 0.38
ALDH1A1 P00352 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691359 0.94 POLB (0.44) NR1I2HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL9691648 0.93 TP53 (0.41) NR1I2MAPTKDM4EGAAPOLB
SCHEMBL9691692 0.92 KMT2A (0.43) HTR1ASLC6A2SLC6A4SLC6A3LMNA
SCHEMBL10914095 0.91 POLB (0.46) NR1I2HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL9691796 0.91 HTR6 (0.43) NR1I2LMNAKDM4EL3MBTL1GAA
SCHEMBL10647671 0.89 NR1I2 (0.39) NR1I2HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL9690850 0.88 GAA (0.40) NR1I2MAPTKDM4EGAAPOLB
SCHEMBL9690807 0.88 POLB (0.44) NR1I2HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL10647063 0.87 POLB (0.43) NR1I2HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL9690877 0.87 HTR6 (0.43) NR1I2HTR1ASLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed