SCHEMBL9691648

SCHEMBL9691648

COC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1ccc(C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
KDM4E B2RXH2 3/20 0.41
GAA P10253 1/20 0.41
NR1I2 O75469 1/20 0.40
SLC1A5 Q15758 1/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SIRT1 Q96EB6 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
RXRA P19793 2/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
BRD4 O60885 1/20 0.38
ATM Q13315 1/20 0.37
KMT2A Q03164 2/20 0.37
HTT P42858 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9691359 0.95 POLB (0.44) TP53KDM4EGAANR1I2POLB
SCHEMBL10814309 0.94 TP53 (0.45) TP53KDM4EGAASLC1A5POLB
SCHEMBL9691625 0.93 NR1I2 (0.42) KDM4EGAANR1I2SLC1A5POLB
SCHEMBL9691661 0.93 TP53 (0.43) TP53KDM4EGAANR1I2SLC1A5
SCHEMBL10914095 0.92 POLB (0.46) TP53KDM4EGAANR1I2POLB
SCHEMBL9691675 0.91 TP53 (0.40) TP53KDM4EGAANR1I2SLC1A5
SCHEMBL9690850 0.91 GAA (0.40) KDM4EGAANR1I2POLBSMN1; SMN2
SCHEMBL9690807 0.91 POLB (0.44) TP53KDM4EGAANR1I2POLB
SCHEMBL10818189 0.90 TP53 (0.41) TP53KDM4EGAANR1I2SLC1A5
SCHEMBL9691403 0.89 TP53 (0.40) TP53KDM4EGAASLC1A5POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed