SCHEMBL9691830

SCHEMBL9691830

COC(=O)OC1=C(C)NC(C)=C(OC(=O)OCCC#N)C1c1ccccc1OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
KDM4E B2RXH2 4/20 0.38
GAA P10253 1/20 0.38
NR1I2 O75469 1/20 0.37
BRD4 O60885 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
HTT P42858 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
SGMS2 Q8NHU3 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689513 0.95 TP53 (0.40) SMN1; SMN2TP53POLBKDM4EGAA
SCHEMBL10914095 0.89 POLB (0.46) SMN1; SMN2TP53POLBKMT2AMEN1
SCHEMBL11303089 0.88 ALDH1A1 (0.48) SMN1; SMN2TP53POLBKMT2AMEN1
SCHEMBL9691359 0.86 POLB (0.44) SMN1; SMN2TP53POLBKMT2AMEN1
SCHEMBL10647063 0.85 POLB (0.43) SMN1; SMN2TP53POLBKMT2AMEN1
SCHEMBL9690807 0.84 POLB (0.44) SMN1; SMN2TP53POLBKMT2AMEN1
SCHEMBL10647317 0.84 POLB (0.42) SMN1; SMN2TP53POLBKMT2AMEN1
SCHEMBL11003624 0.83 KDM4E (0.52) TP53KDM4EGAANR1I2
SCHEMBL10647279 0.82 NPC1 (0.43) SMN1; SMN2POLBKMT2AMEN1KDM4E
SCHEMBL10645304 0.82 POLB (0.41) SMN1; SMN2TP53POLBKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed