SCHEMBL9695753

SCHEMBL9695753

COc1ccc(-c2nnc(C(=O)N(C)C)nc2-c2ccc(OC)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.49
ALDH1A1 P00352 4/20 0.49
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX12 P18054 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
ATR Q13535 1/20 0.42
TSPO P30536 1/20 0.42
MAPT P10636 3/20 0.41
TP53 P04637 3/20 0.41
PTGS2 P35354 1/20 0.41
MGLL Q99685 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9695395 0.77 POLB (0.56) PTGESALDH1A1KDM4EL3MBTL1HTT
SCHEMBL9694185 0.77 RAD52 (0.56) PTGESALDH1A1KDM4EMAPTTP53
Hydrochloric Acid SCHEMBL9694192 0.75 ALDH1A1 (0.61) PTGESALDH1A1NPSR1KDM4ETDP1
SCHEMBL11742743 0.73 ALDH1A1 (0.49) PTGESALDH1A1NPSR1KDM4ELMNA
SCHEMBL1305249 0.73 ALDH1A1 (0.51) PTGESALDH1A1NPSR1KDM4ELMNA
SCHEMBL9548089 0.72 ALDH1A1 (0.58) ALDH1A1KDM4ELMNATDP1L3MBTL1
SCHEMBL21852751 0.71 ALDH1A1 (0.67) ALDH1A1NPSR1KDM4ELMNATDP1
Hydrochloric Acid SCHEMBL9695711 0.71 KDM4E (0.47) ALDH1A1KDM4ETDP1CYP3A4CYP2C9
Anitrazafen SCHEMBL43419 0.71 ALDH1A1 (0.53) PTGESALDH1A1NPSR1KDM4ELMNA
SCHEMBL1305539 0.71 ALDH1A1 (0.56) PTGESALDH1A1NPSR1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992002513-A1 HETEROCYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-02-20 WO disclosed