SCHEMBL9696702

SCHEMBL9696702

Cc1nc2n(c(=O)c1CCN1CCC(C(O)c3nc4cccnc4n3Cc3ccco3)CC1)CCS2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 1/20 0.36
DRD2 P14416 6/20 0.34
HTR1A P08908 6/20 0.34
HTR2A P28223 6/20 0.34
POLB P06746 4/20 0.34
ALDH1A1 P00352 5/20 0.33
TSHR P16473 3/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 2/20 0.33
NPC1 O15118 1/20 0.33
USP2 O75604 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HPGD P15428 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535132 0.85 SLC6A9 (0.43) DRD2HTR1AHTR2APOLBALDH1A1
SCHEMBL9695634 0.78 HPGD (0.42) CACNA2D1HTR1APOLBALDH1A1TSHR
SCHEMBL9537833 0.76 ALDH1A1 (0.39) DRD2HTR1AHTR2APOLBALDH1A1
SCHEMBL9537922 0.72 ALDH1A1 (0.38) DRD2HTR1AHTR2APOLBALDH1A1
SCHEMBL6523129 0.72 HTR2A (0.53) DRD2HTR1AHTR2AALDH1A1TSHR
SCHEMBL6523131 0.72 HTR2A (0.53) DRD2HTR1AHTR2AALDH1A1TSHR
SCHEMBL6523137 0.72 HTR2A (0.53) DRD2HTR1AHTR2AALDH1A1TSHR
Barmastine SCHEMBL30712053 0.70 KDM4E (0.45) DRD2HTR1AHTR2APOLBALDH1A1
Barmastine SCHEMBL141926 0.70 KDM4E (0.45) DRD2HTR1AHTR2APOLBALDH1A1
SCHEMBL9695625 0.70 HRH1 (0.48) HTR2AALDH1A1TSHRLMNAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006086-A1 NOVEL 4-PIPERIDINYLCARBONYL DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-16 WO disclosed