SCHEMBL9696913

SCHEMBL9696913

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SC[S+](C)[O-])[C@H](C)[C@H]12

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.47
PTGS1 P23219 2/20 0.47
ESR1 P03372 2/20 0.47
PDE4A P27815 1/20 0.47
ABCC2 Q92887 1/20 0.42
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
FAP Q12884 1/20 0.35
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CHRM1 P11229 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
SLC29A1 Q99808 1/20 0.32
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10440528 0.84 CACNA1C (0.51) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL9696440 0.82 ESR1 (0.43) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL9696611 0.82 CACNA1C (0.49) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL21580502 0.82 CACNA1C (0.49) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL25519544 0.82 CACNA1C (0.49) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL9695344 0.82 ESR1 (0.44) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL23635213 0.81 CACNA1C (0.48) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL23635250 0.81 CACNA1C (0.48) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL21081298 0.81 CACNA1C (0.48) CACNA1CPTGS1ESR1PDE4AABCC2
SCHEMBL23635249 0.81 CACNA1C (0.48) CACNA1CPTGS1ESR1PDE4AABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US claimed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP claimed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP disclosed