SCHEMBL9696440

SCHEMBL9696440

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SC[S+]([O-])c3ccc(Cl)cc3)[C@H](C)[C@H]12

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
PTGS1 P23219 1/20 0.43
PDE4A P27815 1/20 0.43
CACNA1C Q13936 1/20 0.42
ABCC2 Q92887 1/20 0.39
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
FAP Q12884 1/20 0.32
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9695344 0.86 ESR1 (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696913 0.82 CACNA1C (0.47) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9695126 0.82 CACNA1C (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9738966 0.82 CACNA1C (0.44) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL8437702 0.80 PTGS1 (0.39) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9126535 0.80 PTGS1 (0.39) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10765227 0.77 ABCC2 (0.43) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL9696611 0.77 CACNA1C (0.49) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10440528 0.77 CACNA1C (0.51) ESR1PTGS1PDE4ACACNA1CABCC2
SCHEMBL10440288 0.75 ESR1 (0.48) ESR1PTGS1PDE4ACACNA1CABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US claimed
EP-0481511-A2 Antibiotic C-3 dithioacetal-substituted carbapenem compounds, compositions, and use thereof Bristol-Myers Squibb Company (US) 1992-04-22 EP claimed
US-5116833-A ANTIBIOTIC C-3 DITHIOACETAL-SUBSTITUTED CARBAPENEM COMPOUNDS, COMPOSITIONS, AND METHODS OF USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 1992-05-26 US disclosed