SCHEMBL9698405

SCHEMBL9698405

CC(Cc1ccnc2ccccc12)(NC(=O)O)C(=O)NC(CO)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPK1 P28482 2/20 0.43
CYP3A4 P08684 1/20 0.43
PARP1 P09874 1/20 0.42
PARP3 Q9Y6F1 1/20 0.42
ROCK2 O75116 3/20 0.40
ROCK1 Q13464 3/20 0.40
RPS6KA5 O75582 1/20 0.40
RPS6KA4 O75676 1/20 0.40
PRKACA P17612 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
IRAK1 P51617 1/20 0.40
PRKX P51817 1/20 0.40
PRKG1 Q13976 1/20 0.40
PKN2 Q16513 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540182 0.83 KDM4E (0.41) KDM4EKMT2ATACR1
SCHEMBL7668995 0.82 MAPK1 (0.45) MAPTKMT2AMAPK1CYP3A4ROCK2
SCHEMBL6888621 0.81 TACR1 (0.58) TACR1
SCHEMBL8829867 0.81 TACR1 (0.58) TACR1
SCHEMBL8829871 0.81 TACR1 (0.58) TACR1
SCHEMBL9399753 0.80 CYP3A4 (0.45) MAPK1CYP3A4ROCK2ROCK1RPS6KA5
SCHEMBL9699591 0.80 CCKBR (0.43)
SCHEMBL7669792 0.79 CCKBR (0.52) MAPT
SCHEMBL7663084 0.78 CYP3A4 (0.41) MAPK1CYP3A4PARP1PARP3ROCK2
SCHEMBL9699633 0.78 MAPK1 (0.47) KDM4EMEN1MAPTKMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992004025-A1 AMINO ACID ANALOGS AS CCK ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1992-03-19 WO claimed