SCHEMBL9540182

SCHEMBL9540182

CCCCCCCCC(C)OC(=O)NC(C)(Cc1ccnc2ccccc12)C(=O)NC(CO)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CTSK P43235 2/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSH P09668 1/20 0.40
TACR3 P29371 4/20 0.38
TACR1 P25103 1/20 0.37
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540664 0.85 TACR1 (0.55) TACR3TACR1
SCHEMBL9540669 0.85 TACR1 (0.55) TACR3TACR1
SCHEMBL9538450 0.84 KDM4E (0.42) KDM4EKMT2AL3MBTL1CTSKCTSL
SCHEMBL9698405 0.83 KDM4E (0.45) KDM4EKMT2ATACR1
SCHEMBL9538882 0.80 GABRA1 (0.41) KDM4EKMT2AL3MBTL1TACR3TACR1
SCHEMBL9540187 0.78 PARP1 (0.35) KDM4EKMT2ACTSKCTSLCTSB
SCHEMBL9538034 0.75 TACR3 (0.54) TACR3TACR1
SCHEMBL9338635 0.74 TACR1 (0.55) TACR3TACR1
SCHEMBL9699591 0.74 CCKBR (0.43)
SCHEMBL9539374 0.69 TACR3 (0.45) KDM4EKMT2AL3MBTL1TACR3TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed