SCHEMBL9699255

SCHEMBL9699255

CCN(CC)CC1Cn2c(C)c(Sc3ccccc3)c3cccc(c32)O1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.33
AKR1B1 P15121 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
GBA1 P04062 1/20 0.31
LMNA P02545 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
MEN1 O00255 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700447 0.85 PTGDR2 (0.34) SLC6A4AKR1B1PTGDR2
SCHEMBL9699053 0.83 CASR (0.35) SLC6A4AKR1B1PTGDR2
SCHEMBL9701354 0.81 ADRA2A (0.41)
SCHEMBL9701452 0.81 ADRA2A (0.44)
SCHEMBL9700258 0.80 ADRA2A (0.46)
SCHEMBL9701663 0.80 HRH3 (0.41)
SCHEMBL9700246 0.79 HTR1A (0.34) GBA1
SCHEMBL10471317 0.77 HRH3 (0.39)
SCHEMBL9700627 0.76 HRH3 (0.38)
SCHEMBL9700429 0.76 CNR2 (0.38) SLC6A4AKR1B1PTGDR2LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed