SCHEMBL9699535

SCHEMBL9699535

CCCOCc1cc(O)c(O)c(C(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.43
HMGB1 P09429 1/20 0.42
CXCL12 P48061 1/20 0.42
KAT8 Q9H7Z6 2/20 0.40
PTPN1 P18031 5/20 0.40
RARA P10276 1/20 0.39
RARB P10826 1/20 0.39
TP53 P04637 1/20 0.39
LCK P06239 1/20 0.38
KLKB1 P03952 1/20 0.38
CTSB P07858 1/20 0.38
MMP9 P14780 1/20 0.38
DNMT1 P26358 1/20 0.38
DNMT3B Q9UBC3 1/20 0.38
DNMT3L Q9UJW3 1/20 0.38
DNMT3A Q9Y6K1 1/20 0.38
MCL1 Q07820 1/20 0.37
CA12 O43570 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699529 0.87 HMGB1 (0.45) PPARAHMGB1CXCL12KAT8PTPN1
SCHEMBL23352166 0.84 TP53 (0.47) PPARAHMGB1CXCL12PTPN1TP53
SCHEMBL23750682 0.83 PTPN1 (0.47) PTPN1ALDH1A1ESR1
SCHEMBL9700693 0.80 PRKCE (0.47) PPARAHMGB1CXCL12PTPN1TP53
SCHEMBL22529565 0.78 MCL1 (0.53) PPARAHMGB1CXCL12KAT8PTPN1
SCHEMBL7516702 0.78 RARB (0.51) PPARARARARARBMCL1
SCHEMBL9700687 0.78 HMGB1 (0.52) PPARAHMGB1CXCL12KAT8PTPN1
SCHEMBL27639291 0.77 CYP3A4 (0.53) PTPN1MCL1ALDH1A1PTPN2
SCHEMBL9701888 0.76 HMGB1 (0.44) PPARAHMGB1CXCL12PTPN1LCK
SCHEMBL5676629 0.76 PPARA (0.62) PPARAHMGB1CXCL12KAT8RARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166060-A Prepared by the action of 2,3-dihydroxybenzoate-3,4-dioxygenase on 2,3-dihydroxybenzoic acid CELGENE CORPORATION (US) 1992-11-24 US claimed
EP-0390102-A2 Process for the preparation of pyridine-2,3-dicarboxylic acids CELGENE CORPORATION (US) 1990-10-03 EP claimed
US-5166060-A Prepared by the action of 2,3-dihydroxybenzoate-3,4-dioxygenase on 2,3-dihydroxybenzoic acid CELGENE CORPORATION (US) 1992-11-24 US disclosed
EP-0390102-A2 Process for the preparation of pyridine-2,3-dicarboxylic acids CELGENE CORPORATION (US) 1990-10-03 EP disclosed