SCHEMBL9700693

SCHEMBL9700693

COCc1cc(O)c(O)c(C(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCE Q02156 3/20 0.47
HMGB1 P09429 1/20 0.47
CXCL12 P48061 1/20 0.47
PTPN1 P18031 4/20 0.43
LCK P06239 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MYLK Q15746 2/20 0.42
MEN1 O00255 1/20 0.42
PRKCG P05129 1/20 0.42
MAPT P10636 1/20 0.42
PRKCA P17252 1/20 0.42
APEX1 P27695 1/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KLKB1 P03952 1/20 0.42
CTSB P07858 1/20 0.42
MMP9 P14780 1/20 0.42
DNMT1 P26358 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699529 0.83 HMGB1 (0.45) HMGB1CXCL12PTPN1LCKALDH1A1
SCHEMBL28544278 0.83 AKR1C2 (0.53) HMGB1CXCL12PTPN1ALDH1A1MEN1
SCHEMBL6618063 0.82 PPARA (0.55) PTPN1LCKALDH1A1MEN1MAPT
SCHEMBL9701888 0.81 HMGB1 (0.44) HMGB1CXCL12PTPN1LCKALDH1A1
SCHEMBL24614011 0.80 PRKCE (0.54) PRKCEALDH1A1MYLKMEN1PRKCG
SCHEMBL9699535 0.80 PPARA (0.43) HMGB1CXCL12PTPN1LCKALDH1A1
SCHEMBL9700687 0.79 HMGB1 (0.52) HMGB1CXCL12PTPN1LCKALDH1A1
SCHEMBL28543806 0.79 KLKB1 (0.65) PTPN1LCKKDM4CALDH1A1MEN1
SCHEMBL22529565 0.76 MCL1 (0.53) HMGB1CXCL12PTPN1LCKKLKB1
SCHEMBL18341497 0.76 NPC1 (0.53) ALDH1A1MAPTRECQLKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166060-A Prepared by the action of 2,3-dihydroxybenzoate-3,4-dioxygenase on 2,3-dihydroxybenzoic acid CELGENE CORPORATION (US) 1992-11-24 US claimed
EP-0390102-A2 Process for the preparation of pyridine-2,3-dicarboxylic acids CELGENE CORPORATION (US) 1990-10-03 EP claimed
US-5166060-A Prepared by the action of 2,3-dihydroxybenzoate-3,4-dioxygenase on 2,3-dihydroxybenzoic acid CELGENE CORPORATION (US) 1992-11-24 US disclosed
EP-0390102-A2 Process for the preparation of pyridine-2,3-dicarboxylic acids CELGENE CORPORATION (US) 1990-10-03 EP disclosed