SCHEMBL969974

SCHEMBL969974

OC[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@@H]1OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.51
PDE4D Q08499 1/20 0.46
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
TACR2 P21452 1/20 0.43
PDPK1 O15530 2/20 0.43
MTOR P42345 1/20 0.43
LGALS8 O00214 1/20 0.42
HRAS P01112 2/20 0.40
SLC5A2 P31639 2/20 0.40
BCHE P06276 1/20 0.39
GJB2 P29033 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6659183 1.00 SLC6A2 (0.51) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL969972 1.00 SLC6A2 (0.51) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL630301 1.00 SLC6A2 (0.51) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL8960128 0.95 SLC6A2 (0.52) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL8960525 0.95 SLC6A2 (0.52) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL8960125 0.95 SLC6A2 (0.52) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL8960350 0.95 SLC6A2 (0.52) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL8960222 0.95 SLC6A2 (0.52) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL8960215 0.95 SLC6A2 (0.52) SLC6A2PDE4DTSHRCYP2C19TACR2
SCHEMBL6552387 0.92 SLC6A2 (0.50) SLC6A2PDE4DTSHRCYP2C19TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730601-B1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTIONS UNIV WASHINGTON (US) 2004-07-14 EP claimed
US-9149489-B2 Inhibitors of glycolysis useful in the treatment of brain tumors BOARD OF REGENTS, UNIVERSITY OF TEXAS SYSTEM (US) 2015-10-06 US disclosed
US-20110003758-A1 Inhibitors of Glycolysis Useful In the Treatment of Brain Tumors NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-01-06 US disclosed
WO-2009108926-A1 INHIBITORS OF GLYCOLYSIS USEFUL IN THE TREATMENT OF BRAIN TUMORS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2009-09-03 WO disclosed
US-5491152-A Derivatives of cyclic ethers and sulfides for the treatment of atherosclerosis THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-02-13 US disclosed
WO-1995014028-A9 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFECTIONS 1995-08-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110003758-A1 Inhibitors of Glycolysis Useful In the Treatment of Brain Tumors PDK2, G6PD, PCK2 SLC6A2 1422/4885PDE4D 2963/4885TSHR 3744/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.