SCHEMBL9700186

SCHEMBL9700186

CCCCCC#Cc1cccc(C=O)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.45
FFAR1 O14842 2/20 0.44
FFAR4 Q5NUL3 1/20 0.42
MMP2 P08253 1/20 0.41
MMP12 P39900 1/20 0.41
MAPT P10636 3/20 0.39
GGPS1 O95749 1/20 0.38
MAPK1 P28482 1/20 0.37
GPR84 Q9NQS5 1/20 0.37
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
GRM5 P41594 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP2D6 P10635 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1852576 0.98 KCNH2 (0.48) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL8846088 0.98 KCNH2 (0.48) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL7680519 0.98 KCNH2 (0.48) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL10795164 0.98 KCNH2 (0.48) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL493774 0.95 FFAR1 (0.45) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL9559955 0.88 FFAR1 (0.52) FFAR1FFAR4MAPTCYP3A4TSHR
SCHEMBL2233459 0.81 FFAR1 (0.52) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL10752111 0.80 FFAR1 (0.47) KCNH2FFAR1FFAR4MMP2MMP12
SCHEMBL3899508 0.80 FFAR1 (0.50) FFAR1ALDH1A1
SCHEMBL30688451 0.80 FFAR1 (0.50) FFAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503079-A1 PYRIDAZINONE-SUBSTITUTED ETHYNYLPHENYL DERIVATIVE AND REMEDY FOR CIRCULATORY ORGAN DISEASE CONTAINING THE SAME AS ACTIVE INGREDIENT KAKEN PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed