SCHEMBL9700347

SCHEMBL9700347

CC(=O)CC(=O)c1ccc([S+](C)[O-])cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.39
KMT2A Q03164 3/20 0.39
NPC1 O15118 3/20 0.39
MEN1 O00255 2/20 0.39
ERCC5 P28715 4/20 0.38
FEN1 P39748 4/20 0.38
MAPT P10636 3/20 0.38
ALOX15 P16050 2/20 0.38
MAPK1 P28482 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
CES1 P23141 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTPN1 P18031 2/20 0.37
HAO1 Q9UJM8 5/20 0.37
ALDH1A1 P00352 3/20 0.36
TP53 P04637 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700437 0.82 SMN1; SMN2 (0.44) RAB9AKMT2ANPC1MEN1KDM4E
SCHEMBL2003577 0.82 KMT2A (0.52) RAB9AKMT2ANPC1MEN1ERCC5
SCHEMBL31185587 0.81 SMN1; SMN2 (0.50) RAB9AKMT2ANPC1MEN1MAPT
SCHEMBL10830356 0.79 GSK3B (0.53) RAB9AERCC5FEN1MAPTMAPK1
SCHEMBL1535161 0.79 GSK3B (0.57) PTPN1GSK3B
SCHEMBL31256698 0.78 MAPK1 (0.47) RAB9AKMT2ANPC1MAPTMAPK1
SCHEMBL27719499 0.76 HSD17B3 (0.39) RAB9AKMT2ANPC1TDP1KDM4E
SCHEMBL17907433 0.76 ALDH1A1 (0.48) RAB9ANPC1MAPTMAPK1HPGD
SCHEMBL11681650 0.75 HSD17B3 (0.61) RAB9ANPC1HPGDSMN1; SMN2
SCHEMBL3035986 0.74 NPC1 (0.67) RAB9AKMT2ANPC1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed