SCHEMBL9700512

SCHEMBL9700512

O=C(O)c1cn(C2CC2)c2c(F)c(-n3ccnc3)c(F)cc2c1=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 6/20 0.64
TOP2B Q02880 6/20 0.64
KCNH2 Q12809 5/20 0.53
ALDH1A1 P00352 4/20 0.52
POLB P06746 2/20 0.52
OPRM1 P35372 2/20 0.52
CHRM2 P08172 1/20 0.52
CHRM1 P11229 1/20 0.52
OPRD1 P41143 1/20 0.52
KDM4E B2RXH2 3/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 2/20 0.50
PRKD3 O94806 1/20 0.50
ALOX15 P16050 1/20 0.50
CLK2 P49760 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
GSK3B P49841 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10875605 0.90 TOP2A (0.56) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL10875166 0.90 ALDH1A1 (0.62) TOP2ATOP2BKCNH2ALDH1A1POLB
Hydrochloric Acid SCHEMBL9773808 0.89 KCNH2 (0.61) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL10876273 0.87 TOP2A (0.48) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL9519028 0.84 TOP2A (0.64) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL10679827 0.83 MEN1 (0.61) TOP2ATOP2BKCNH2POLBMEN1
SCHEMBL10849002 0.82 LMNA (0.66) TOP2ATOP2BKCNH2ALDH1A1POLB
Hydrochloric Acid SCHEMBL10850221 0.82 LMNA (0.65) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL9270913 0.81 KCNH2 (0.53) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL10881020 0.81 KDM4E (0.56) TOP2ATOP2BALDH1A1POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098913-A Bactericides for grampositive bacteria LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 1992-03-24 US disclosed
EP-0203488-A2 7-Azolyl-1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids and 1,8-naphthyridine carboxylic acids, process for their preparation and bactericidal agents containing them BAYER AG (DE) 1986-12-03 EP disclosed