SCHEMBL9700820

SCHEMBL9700820

Cc1cn(-c2ccc(N)c(CO)c2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP19A1 P11511 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NR2E1 Q9Y466 4/20 0.43
CYP2E1 P05181 1/20 0.41
CYP2A6 P11509 1/20 0.41
MAOA P21397 4/20 0.40
MAOB P27338 4/20 0.40
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
NOTUM Q6P988 1/20 0.35
WNT3A P56704 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1824196 0.87 CYP3A4 (0.46) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
Hydrochloric Acid SCHEMBL1823628 0.85 CYP3A4 (0.44) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL9740148 0.84 CYP3A4 (0.43) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL9740152 0.83 CYP3A4 (0.46) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL28949276 0.82 NOTUM (0.46) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL15442444 0.81 NR2E1 (0.49) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL9701793 0.80 NR2E1 (0.48) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL9701824 0.79 NR2E1 (0.46) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL3343040 0.76 NR2E1 (0.48) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL30217888 0.75 IP6K1 (0.49) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5171851-A Cardiac stimulant DONG-A PHARM. CO., LTD. (KR) 1992-12-15 US disclosed
EP-0510235-A1 Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same DONG-A PHARM. CO., LTD. (KR) 1992-10-28 EP disclosed