SCHEMBL9701793

SCHEMBL9701793

Cc1cn(-c2ccc(N)c(C)c2)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 1/20 0.48
CYP3A4 P08684 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP19A1 P11511 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP2E1 P05181 1/20 0.46
CYP2A6 P11509 1/20 0.46
RAD52 P43351 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
MAOA P21397 4/20 0.45
MAOB P27338 4/20 0.45
GAA P10253 2/20 0.41
THRB P10828 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15442444 0.88 NR2E1 (0.49) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL3343040 0.86 NR2E1 (0.48) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL1824196 0.81 CYP3A4 (0.46) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL15222204 0.81 MAOA (0.50) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL1828556 0.80 NR2E1 (0.43) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
Hydrochloric Acid SCHEMBL1823628 0.80 CYP3A4 (0.44) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL9700820 0.80 CYP3A4 (0.44) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL22198918 0.79 CYP1A2 (0.46) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL27985278 0.79 CYP1A2 (0.65) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL30217888 0.79 IP6K1 (0.49) NR2E1CYP3A4CYP1A2CYP2D6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5171851-A Cardiac stimulant DONG-A PHARM. CO., LTD. (KR) 1992-12-15 US disclosed
EP-0510235-A1 Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same DONG-A PHARM. CO., LTD. (KR) 1992-10-28 EP disclosed