SCHEMBL9701104

SCHEMBL9701104

CCOc1cc[c]c(-c2ccncc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
KMT2A Q03164 3/20 0.45
CYP2C9 P11712 2/20 0.45
MEN1 O00255 2/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 1/20 0.45
CYP1A2 P05177 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
S1PR1 P21453 5/20 0.44
NPSR1 Q6W5P4 1/20 0.41
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
CYP19A1 P11511 2/20 0.39
CYP11B1 P15538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700067 0.88 CYP2D6 (0.49) CYP3A4CYP2D6CYP2C9KDM4EALDH1A1
SCHEMBL8532102 0.85 NQO1 (0.50) CYP3A4CYP2D6KMT2ACYP2C9MEN1
SCHEMBL6194180 0.83 TTK (0.43) CYP3A4KDM4EALDH1A1NPC1HPGD
SCHEMBL15067112 0.82 NQO1 (0.48) CYP3A4CYP2D6KMT2AMEN1KDM4E
SCHEMBL17536735 0.82 MAPT (0.39) CYP3A4KMT2AKDM4EALDH1A1HPGD
SCHEMBL9698295 0.81 PDGFRB (0.46) CYP3A4CYP2D6KMT2ACYP2C9MEN1
SCHEMBL9559856 0.81 CHRNA7 (0.41) CYP3A4CYP2D6CYP1A2CYP2C19HSD17B10
SCHEMBL6382918 0.81 CYP11B1 (0.44) KMT2AKDM4EALDH1A1NPC1HPGD
SCHEMBL2222934 0.78 NQO1 (0.42) CYP3A4CYP2D6CYP2C9KDM4EALDH1A1
SCHEMBL9293790 0.78 EPHX2 (0.38) CYP3A4CYP2C9CYP2C19SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145858-A Antiinflammatory SMITHKLINE BEECHAM CORP. (US) 1992-09-08 US disclosed
US-5002941-A Antiarthritic agents, arachidonic acid metabolism SMITHKLINE BEECHAM CORPORATION (US) 1991-03-26 US disclosed