SCHEMBL9700067

SCHEMBL9700067

CCCOc1cc[c]c(-c2ccncc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.49
CYP3A4 P08684 2/20 0.49
KDM4E B2RXH2 3/20 0.48
NPC1 O15118 2/20 0.48
ALDH1A1 P00352 2/20 0.48
RAB9A P51151 2/20 0.48
HSD17B10 Q99714 2/20 0.48
HPGD P15428 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
S1PR1 P21453 1/20 0.44
S1PR3 Q99500 1/20 0.44
ROCK1 Q13464 4/20 0.42
ROCK2 O75116 3/20 0.42
CYP2C9 P11712 3/20 0.42
MAPT P10636 4/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
DYRK3 O43781 1/20 0.40
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701104 0.88 CYP3A4 (0.45) CYP2D6CYP3A4KDM4ENPC1ALDH1A1
SCHEMBL15066586 0.84 KMT2A (0.42) KDM4EMAPTTSHR
SCHEMBL7078066 0.82 LTA4H (0.50) NPC1ALDH1A1RAB9AMAPTTSHR
SCHEMBL2222934 0.82 NQO1 (0.42) CYP2D6CYP3A4KDM4ENPC1ALDH1A1
SCHEMBL8300230 0.81 CYP1A1 (0.41) CYP2D6KDM4ENPC1ALDH1A1RAB9A
SCHEMBL9698295 0.79 PDGFRB (0.46) CYP2D6CYP3A4KDM4ENPC1ALDH1A1
SCHEMBL8187884 0.78 ALDH1A1 (0.39) CYP2D6KDM4ENPC1ALDH1A1RAB9A
SCHEMBL8007736 0.77 CYP19A1 (0.48) CYP2D6CYP3A4NPC1RAB9AHSD17B10
SCHEMBL9783835 0.76 NR5A1 (0.50) CYP2D6CYP3A4KDM4EALDH1A1HPGD
SCHEMBL15067951 0.75 LTA4H (0.44) CYP2D6CYP3A4NPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145858-A Antiinflammatory SMITHKLINE BEECHAM CORP. (US) 1992-09-08 US disclosed
US-5002941-A Antiarthritic agents, arachidonic acid metabolism SMITHKLINE BEECHAM CORPORATION (US) 1991-03-26 US disclosed