SCHEMBL9701519

SCHEMBL9701519

O=C(O)Cn1cc(Cc2ccccc2)c2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.60
HDAC1 Q13547 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
HDAC3 O15379 1/20 0.57
HTR6 P50406 3/20 0.57
ALDH1A1 P00352 3/20 0.57
TBXAS1 P24557 1/20 0.56
STAT3 P40763 1/20 0.56
ALOX5 P09917 1/20 0.56
KDM4E B2RXH2 3/20 0.56
KRAS P01116 1/20 0.55
AKR1A1 P14550 3/20 0.54
AKR1B1 P15121 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27691201 0.90 KMT2A (0.56) KMT2AHDAC1HDAC8HDAC6HDAC3
SCHEMBL1520240 0.85 TBXAS1 (0.64) KMT2AALDH1A1TBXAS1STAT3ALOX5
SCHEMBL18180209 0.84 CDC25A (0.63) KMT2AALDH1A1TBXAS1STAT3KDM4E
SCHEMBL12874520 0.84 KMT2A (0.66) KMT2AALDH1A1TBXAS1STAT3ALOX5
SCHEMBL421164 0.83 KMT2A (0.52) KMT2AALDH1A1TBXAS1ALOX5AKR1A1
SCHEMBL6567317 0.83 ALDH1A1 (0.58) KMT2AHTR6ALDH1A1TBXAS1STAT3
SCHEMBL8021536 0.81 MCL1 (0.60) KMT2AHTR6ALDH1A1TBXAS1STAT3
SCHEMBL27915317 0.81 CNR2 (0.51) KMT2AHDAC1HDAC8HDAC6ALDH1A1
SCHEMBL27711191 0.81 TP53 (0.57) KMT2AALDH1A1STAT3KDM4EAKR1A1
SCHEMBL27691209 0.81 KMT2A (0.50) KMT2AHDAC1HDAC8HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132319-A Antiasthmatic, antiinflammatory, antiallergen and cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1992-07-21 US disclosed