SCHEMBL9701949

SCHEMBL9701949

C=C=C(CN)c1ccc(OC)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.54
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
CA7 P43166 1/20 0.47
TPMT P51580 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
ELANE P08246 1/20 0.47
PRSS1 P07477 4/20 0.46
MAPK1 P28482 1/20 0.46
PDE4A P27815 3/20 0.45
PDE4B Q07343 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703287 0.77 CA1 (0.46) CA1CA2PRSS1ALDH1A1MAPT
SCHEMBL14611953 0.77 MAOB (0.58) MAOBCYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL9701899 0.75 PARP1 (0.51) TSHRPRSS1MAPK1PDE4APDE4B
SCHEMBL9701879 0.74 MAPT (0.47) CYP2C19CYP1A2TSHRCA12CA1
SCHEMBL9700914 0.74 ALDH1A1 (0.41) TSHRPDE4APDE4BPDE4CPDE4D
SCHEMBL1260548 0.74 TSHR (0.63) MAOBCYP2C9CYP2C19CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL4512041 0.72 TSHR (0.61) MAOBCYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL9703267 0.72 CA12 (0.44) CYP3A4CA12CA1CA2CA4
Hydrochloric Acid SCHEMBL29112504 0.72 TSHR (0.61) MAOBCYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL18848298 0.72 CYP2C9 (0.61) MAOBCYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120764-A Administering penicillamine and allenylamines to inhibit crosslinking of collagen MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-09 US disclosed
EP-0374440-A2 Inhibitors of lysyl oxidase MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-27 EP disclosed