SCHEMBL9702222

SCHEMBL9702222

CCCc1cc2cccnc2n1Cc1ccc(-c2ccccc2-c2nnnn2C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 7/20 0.57
AGTR2 P50052 7/20 0.57
AGT P01019 2/20 0.47
PPARG P37231 2/20 0.43
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
P2RX7 Q99572 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701476 0.87 AGTR1 (0.54) AGTR1AGTR2AGTPPARG
SCHEMBL9851487 0.84 AGTR1 (0.63) AGTR1AGTR2AGTPPARG
SCHEMBL9259102 0.84 AGTR1 (0.54) AGTR1AGTR2AGT
SCHEMBL9851410 0.82 AGTR1 (0.64) AGTR1AGTR2AGTPPARG
SCHEMBL9854421 0.81 AGTR1 (0.62) AGTR1AGTR2AGT
SCHEMBL9263837 0.81 AGT (0.57) AGTR1AGTR2AGT
SCHEMBL9851456 0.81 AGTR1 (0.52) AGTR1AGTR2AGTP2RX7
SCHEMBL9851481 0.81 AGTR1 (0.54) AGTR1AGTR2AGT
SCHEMBL7012281 0.79 AGTR1 (0.53) AGTR1AGTR2AGTPPARG
SCHEMBL9265478 0.79 AGTR1 (0.56) AGTR1AGTR2AGTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497516-A1 Substituted pyrrolo-fused 6-membered heterocycles as angiotensin II antagonists MERCK & CO. INC. (US) 1992-08-05 EP disclosed
US-5124335-A Hypotensive agents, antiglaucoma agents MERCK & CO., INC. (US) 1992-06-23 US disclosed