SCHEMBL9702758

SCHEMBL9702758

C=C=C(CN)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
CYP3A4 P08684 2/20 0.36
MAPT P10636 2/20 0.36
BLM P54132 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
F12 P00748 1/20 0.36
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36
PKM P14618 1/20 0.36
POLB P06746 1/20 0.36
PARP1 P09874 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36
PMP22 Q01453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702759 0.80 MAPT (0.41) CYP3A4MAPTBLMTDP1PKM
SCHEMBL9700915 0.78 ALDH1A1 (0.38) HDAC1TDP1PKMMEN1HPGD
SCHEMBL9702052 0.78 ALDH1A1 (0.46) CYP3A4MAPTTDP1PKMPARP1
SCHEMBL16660765 0.77 PTPN1 (0.46) MAOAMAOBCYP3A4MAPTTDP1
SCHEMBL1173628 0.77 ATM (0.45) MAOAMAOBMAPTBLML3MBTL1
SCHEMBL14000035 0.77 HDAC1 (0.38) HDAC1HDAC2CYP3A4MAPTBLM
SCHEMBL11663847 0.76 POLB (0.35) MAOAMAOBCYP3A4MAPTTDP1
SCHEMBL28357466 0.74 HDAC1 (0.36) HDAC1HDAC2CYP3A4MAPTBLM
SCHEMBL9703287 0.74 CA1 (0.46) HDAC1HDAC2MAPTPARP1CES1
SCHEMBL9701899 0.73 PARP1 (0.51) MAPTPKMPARP1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2180855-A None JP disclosed
US-5120764-A Administering penicillamine and allenylamines to inhibit crosslinking of collagen MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-09 US disclosed
JP-H02180855-A LYSIL OXIDASE INHIBITOR MERRELL DOW PHARMACEUT INC 1990-07-13 JP disclosed
EP-0374440-A2 Inhibitors of lysyl oxidase MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-27 EP disclosed