SCHEMBL9703014

SCHEMBL9703014

CCCC(=O)NNC(=O)c1ccc(OC)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.79
LMNA P02545 2/20 0.79
L3MBTL1 Q9Y468 1/20 0.71
HTT P42858 2/20 0.64
CRHBP P24387 2/20 0.64
CRHR2 Q13324 2/20 0.64
KDM4E B2RXH2 1/20 0.64
PLAU P00749 1/20 0.62
ELANE P08246 1/20 0.62
HDAC3 O15379 1/20 0.61
HDAC1 Q13547 1/20 0.61
HDAC2 Q92769 1/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
GAA P10253 1/20 0.61
CYP2C19 P33261 1/20 0.61
KMT2A Q03164 3/20 0.60
MAPT P10636 1/20 0.59
POLB P06746 1/20 0.58
CTDSP1 Q9GZU7 1/20 0.58
CA1 P00915 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10793129 0.85 ALDH1A1 (0.65) ALDH1A1LMNAL3MBTL1HTTCRHBP
SCHEMBL11705060 0.84 MAPT (0.79) ALDH1A1LMNAL3MBTL1CRHBPCRHR2
SCHEMBL6770004 0.82 LMNA (0.73) ALDH1A1LMNAL3MBTL1HTTCRHBP
SCHEMBL10594113 0.80 ALDH1A1 (0.66) ALDH1A1LMNAL3MBTL1HTTKDM4E
SCHEMBL5673419 0.80 POLB (0.65) ALDH1A1L3MBTL1KDM4ESMN1; SMN2GAA
SCHEMBL4930749 0.78 ALDH1A1 (0.68) ALDH1A1LMNAL3MBTL1HTTCRHBP
SCHEMBL19825010 0.78 MAPT (0.65) ALDH1A1LMNAL3MBTL1HTTCRHBP
SCHEMBL4927732 0.78 GAA (0.75) ALDH1A1LMNAL3MBTL1HTTKDM4E
SCHEMBL4930245 0.78 MAPT (0.69) ALDH1A1LMNAL3MBTL1CRHBPCRHR2
SCHEMBL19899864 0.78 MAPT (0.69) ALDH1A1LMNAL3MBTL1CRHBPCRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5143642-A Thiadiazoles MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-09-01 US disclosed