SCHEMBL9704385

SCHEMBL9704385

CC(=O)NC(C#N)c1cccc(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
ALDH1A1 P00352 3/20 0.43
AKR1C3 P42330 1/20 0.39
AKR1C1 Q04828 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
POLB P06746 1/20 0.37
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9284618 0.88 ALDH1A1 (0.41) CYP1A2ALDH1A1HPGDMAPTHTT
SCHEMBL14065364 0.80 ALDH1A1 (0.53) CYP1A2ALDH1A1AKR1C3AKR1C1POLB
SCHEMBL9704729 0.79 ALDH1A1 (0.38) CYP1A2ALDH1A1AKR1C3AKR1C1MAPT
SCHEMBL7860940 0.79 HPGD (0.40) ALDH1A1HPGDL3MBTL1
SCHEMBL2769652 0.78 ALDH1A1 (0.59) CYP1A2ALDH1A1SMN1; SMN2L3MBTL1POLB
SCHEMBL3881452 0.78 ALDH1A1 (0.59) CYP1A2ALDH1A1SMN1; SMN2L3MBTL1POLB
SCHEMBL12341890 0.78 ALDH1A1 (0.59) CYP1A2ALDH1A1SMN1; SMN2L3MBTL1POLB
SCHEMBL3893098 0.78 ALDH1A1 (0.59) CYP1A2ALDH1A1SMN1; SMN2L3MBTL1POLB
SCHEMBL4175399 0.76 ALDH1A1 (0.40) ALDH1A1AKR1C3AKR1C1NPC1CASP3
SCHEMBL9152220 0.75 PGK1 (0.52) ALDH1A1AKR1C3AKR1C1NPSR1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175153-A Antiischemic agents or antiepileptic agents WARNER-LAMBERT COMPANY (US) 1992-12-29 US disclosed