SCHEMBL9704532

SCHEMBL9704532

Cc1ccnc2c1NC(=O)c1cccnc1N2C(C)C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.62
POLB P06746 2/20 0.62
LMNA P02545 1/20 0.62
ADORA3 P0DMS8 1/20 0.62
MAPK1 P28482 1/20 0.62
ADORA2A P29274 1/20 0.62
ADORA1 P30542 1/20 0.62
PDE3A Q14432 1/20 0.62
DAO P14920 1/20 0.41
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP1A2 P05177 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
MCL1 Q07820 1/20 0.36
TNKS2 Q9H2K2 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6712803 0.83 ALDH1A1 (0.53) ALDH1A1POLBLMNAADORA3MAPK1
SCHEMBL8304745 0.81 CYP1A2 (0.49) ALDH1A1POLBLMNAADORA3MAPK1
SCHEMBL8300618 0.79 ALDH1A1 (0.62) ALDH1A1POLBLMNAADORA3MAPK1
Nevirapine SCHEMBL14031771 0.78 ALDH1A1 (0.82) ALDH1A1POLBLMNAADORA3MAPK1
Nevirapine SCHEMBL29393780 0.77 ALDH1A1 (1.00) ALDH1A1POLBLMNAADORA3MAPK1
Nevirapine SCHEMBL30267890 0.77 ALDH1A1 (1.00) ALDH1A1POLBLMNAADORA3MAPK1
Nevirapine SCHEMBL3232525 0.77 ALDH1A1 (1.00) ALDH1A1POLBLMNAADORA3MAPK1
Nevirapine SCHEMBL3318 0.77 ALDH1A1 (1.00) ALDH1A1POLBLMNAADORA3MAPK1
Nevirapine SCHEMBL29614675 0.77 ALDH1A1 (1.00) ALDH1A1POLBLMNAADORA3MAPK1
SCHEMBL14439913 0.76 LMNA (0.59) ALDH1A1POLBLMNAADORA3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482481-A1 Method for the preparation of 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1992-04-29 EP disclosed