SCHEMBL9705707

SCHEMBL9705707

CN(C)c1nc(F)nc2nc[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.56
PDPK1 O15530 2/20 0.56
CHEK1 O14757 1/20 0.56
AURKA O14965 1/20 0.56
CHEK2 O96017 1/20 0.56
HSP90AA1 P07900 1/20 0.56
HSP90AB1 P08238 1/20 0.56
PRKACA P17612 1/20 0.56
CCNE1 P24864 1/20 0.56
MARK3 P27448 1/20 0.56
RPS6KA3 P51812 1/20 0.56
PRKCD Q05655 1/20 0.56
LRRK2 Q5S007 1/20 0.56
MARK2 Q7KZI7 1/20 0.56
EGFR P00533 1/20 0.40
CSF1R P07333 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAP3K5 Q99683 2/20 0.38
HTT P42858 2/20 0.38
GDA Q9Y2T3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL401117 0.79 PDPK1 (0.59) CDK2PDPK1CHEK1AURKACHEK2
SCHEMBL6747380 0.79 CHEK1 (0.56) CDK2PDPK1CHEK1AURKACHEK2
SCHEMBL4523841 0.78 CDK2 (0.51) CDK2PDPK1CHEK1AURKACHEK2
SCHEMBL11212991 0.76 PDPK1 (0.41) CDK2PDPK1CHEK1AURKACHEK2
SCHEMBL2526552 0.75 PDPK1 (0.44) CDK2PDPK1LRRK2MAP3K5GDA
Dimethyladenine SCHEMBL152594 0.72 LRRK2 (1.00) CDK2PDPK1CHEK1AURKACHEK2
Dimethyladenine SCHEMBL29349831 0.72 LRRK2 (1.00) CDK2PDPK1CHEK1AURKACHEK2
SCHEMBL8851 0.72 PDPK1 (0.66) CDK2PDPK1LRRK2MAP3K5GDA
SCHEMBL356178 0.72 DPP4 (0.61) CDK2PDPK1GDATNNI3KADORA3
SCHEMBL29375265 0.72 PDPK1 (0.66) CDK2PDPK1LRRK2MAP3K5GDA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO disclosed